Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki data for polymerid = 49000903,50004132
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85518(tc-NH2 | trans-cinnamoyl-LIGRLO-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85517(CAS_171436-38-7 | SL-NH2 | SLIGRL-NH2)
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50440869(CHEMBL2431727)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]2-furoyl-LIGRL-NH2 from human PAR2 expressed in human NCTC-2544 cells by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50134199(CHEMBL3735057)
Affinity DataKi:  627nMAssay Description:Displacement of [3H]furoyl-LIGRL-NH2 from human protease-activated receptor 2 in NCTC-2544 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50134200(CHEMBL3735405)
Affinity DataKi:  1.94E+3nMAssay Description:Displacement of [3H]furoyl-LIGRL-NH2 from human protease-activated receptor 2 in NCTC-2544 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85516(CAS_141923-41-3 | P5-NH2 | SFLLR-NH2)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteinase-activated receptor 2(RAT)
The University of Calgary

Curated by PDSP Ki Database
LigandPNGBDBM85088(SFLLR-OH)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed